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The testis has a dual function: spermatogenesis and the production of T The latter takes places in the Leydig cells The daily production of T in adulthood is about 5 7 mg T diffuses passively into cells of the target organs of androgens To exert its biologic action, it must bind to the androgen receptor, though there are also a number of biologic actions of T that do not require receptor activation For some of its biologic actions T is a prohormone After diffusion into the cell, T may be converted to 5 -dihydrotestosterone (DHT) or estradiol There are two types of 5 reductase enzymes that convert T to DHT 5 reductase type 1 is predominantly located in skin, liver, and brain whereas 5 reductase type 2 is almost exclusively distributed in the classical androgendependent organs such as prostate,seminal vesicles, and testicles DHT and T bind to the same androgen receptor, although DHT has an approximately tenfold greater af nity for the receptor and its dissociation is slower, resulting in a considerably higher biopotency than T The conversion of T to DHT can be viewed as an androgen ampli cation mechanism in organs that require a strong androgen action, such as
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Testosterone is a lipophilic molecule and its solubility in blood is limited Only 2% of circulating T is free, non-bound to transport proteins, able to diffuse into cells, and immediately available for biologic action Approximately 60% of circulating T is bound with high af nity to sex hormone binding globulin (SHBG), and 38% is loosely bound and transported by albumin The free fraction of T (FT, 2%) and the albumin-bound fraction ( 38%) have been termed bioavailable testosterone (BT), since these two fractions are readily available for biologic action Testosterone has a high af nity with SHBG and changes in concentrations of circulating SHBG impact on the bioavailability of T SHBG is produced by the liver and a number of conditions and hormones in uence its production Androgens and growth hormone decrease circulating SHBG, which increases BT, and ampli es the action of T along with the combined anabolic effects of growth hormone (GH) and T Andro-
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testosterone CNS, central nervous system; FSH, follicle stimulating hormone; GnRH, gonadotropinreleasing hormone; LH, luteinizing hormone
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roaming Roaming is an IP-based service that deals with the movement of users not subnets or hosts among a set of ISPs that have agreed to cooperate In a roaming scenario, users of an ISP in New Jersey, who only have dial-up accounts, can make a local call to a cooperating ISP s local number while in California The California ISP forwards the authentication request to the home ISP, and, based on the home ISP s response, grants or denies access The remote ISP may also cut accounting records if roaming access is subject to a surcharge Practical roaming services have phone book servers from which roaming users can retrieve lists of local access numbers Even more advanced mobility services, the needs for which are still emerging, include wireless LANs, third-generation wireless, and mobile routers
hroughout this book, we mention various professionals and professional organizations that offer the skills, expertise, and basic information that can help you build a real estate investment portfolio that works Knowing that help is available is one thing knowing when to call on help, and the best source of help in any given situation, is another And, as always, you ll experience situations where a bit of cross-pollination will be more helpful than going straight to the one obvious choice This chapter highlights some of the resources available, the problems they can help you solve, and the ways you can make use of the expertise they offer to develop a successful portfolio
gen de ciency, estrogens, hyperthyroidism, and liver disease increase circulating SHBG, and consequently limit its biologic action SHBG also binds estradiol but with lower af nity than T, such that certain conditions may be associated with signs of estrogen excess such as gynecomastia Overweightness with its associated hyperinsulinism, corticosteroids, and hypothyroidism reduce circulating SHBG and result in low total plasma concentrations
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